Adult

Pyrimethamine

Warning

General Information

Anti-protozoal

Restricted formulary antimicrobial: For details see OUH netFormulary

For all information regarding interactions, contraceptions, pregnancy and breastfeeding and additional information, see BNF

Standard dose

See ocular toxoplasmosis guideline

For other indications, contact micro/ID for advice

Obesity

No data available, use standard dosing.

Renal and hepatic impairment

Renal impairment

No data available, use standard dosing.

Hepatic impairment

Manufacturer advises caution in hepatic impairment

References

  1. British National Formulary. Pyrimethamine. BNF online. Accessed via https://bnf.nice.org.uk/drugs/pyrimethamine/ Accessed 29/05/26.
  2. GlaxoSmithKline UK. Daraprim (pyrimethamine). Summary of Product Characteristics.. Available at: https://www.medicines.org.uk/emc/product/938/smpc#gref Accessed 28/05/26.
  3. Sanfordguide.com. Sanford Guide.  Last updated: 08/05/26. Available at: https://web.sanfordguide.com/en/drug-information/antiparasitic-agents/antimalarials/pyrimethamine Accessed 2/05/26.
  4. The Renal Drug Database. Pentamidine. Last updated 23/09/24. Available at: https://www.renaldrugdatabase.com/s/article/PYRIMETHAMINE 29/05/26.

Editorial Information

Last reviewed: 06 Jul 2026

Next review date: 06 Jul 2029

Author(s): AMST.